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Cyproterone acetate
CAS No. 427-51-0
Cyproterone acetate ( Androcur; CPA; Cyprostat; NSC 81430; SH 714 )
Catalog No. M14450 CAS No. 427-51-0
Cyproterone acetate is an androgen receptor (AR) antagonist with IC50 of 7.1 nM, as well as a weak progesterone receptor agonist with weak pro-gestational and glucocorticoid activity.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | 30 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NameCyproterone acetate
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NoteResearch use only, not for human use.
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Brief DescriptionCyproterone acetate is an androgen receptor (AR) antagonist with IC50 of 7.1 nM, as well as a weak progesterone receptor agonist with weak pro-gestational and glucocorticoid activity.
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DescriptionCyproterone acetate is an androgen receptor (AR) antagonist with IC50 of 7.1 nM, as well as a weak progesterone receptor agonist with weak pro-gestational and glucocorticoid activity.
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SynonymsAndrocur; CPA; Cyprostat; NSC 81430; SH 714
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PathwayEndocrinology/Hormones
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TargetAndrogen Receptor (AR)
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RecptorAndrogen Receptor
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Research AreaEndocrinology
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Indication——
Chemical Information
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CAS Number427-51-0
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Formula Weight416.94
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Molecular FormulaC24H29ClO4
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Purity>98%(HPLC)
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SolubilityEthanol: 10 mg/mL (23.98 mM); DMSO: 83 mg/mL (199.06 mM)
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SMILESCC(O[C@]1(C(C)=O)CC[C@]2([H])[C@]1(C)CC[C@]3([H])[C@@]4(C)[C@](C5)([H])[C@]5([H])C(C=C4C(Cl)=C[C@@]23[H])=O)=O
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Chemical Name(2aR,3aS,3bS,3cS,5aS,6R,8aS,8bR)-6-acetyl-10-chloro-3b,5a-dimethyl-2-oxo-2,2a,3,3a,3b,3c,4,5,5a,6,7,8,8a,8b-tetradecahydrocyclopenta[a]cyclopropa[g]phenanthren-6-yl acetate
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Sonneveld E, et al. Toxicol Sci. 2005, 83(1), 136-148.
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